Publications

Císařová, I.; Formánek, B.; Tauchman, J.; Vesely, J. Access to Spirocyclic Benzothiophenones with Multiple Stereocenters via an Organocatalytic Cascade Reaction. Journal of Organic Chemistry 2020, 85 (13), 8510-8521 DOI: 10.1021/acs.joc.0c00882.

Kamlar, M.; Císařová, I.; Hybelbauerová, S.; Vesely, J. Asymmetric Allylic Amination of Morita-Baylis-Hillman Carbonates with Silylated tert-Butylhydroxycarbamate Derivatives. European Journal of Organic Chemistry 2017, No. 14, 1926-1930 DOI: 10.1002/ejoc.201700222.

Číhalová, S.; Dziedzic, P.; Córdova, A.; Vesely, J. Asymmetric Aza-Morita-Baylis-Hillman-Type Reactions: The Highly Enantioselective Reaction between Unmodified α,β- Unsaturated Aldehydes and N-Acylimines by Organo-co-catalysis. Advanced Synthesis & Catalysis 2011, 353 (7), 1096-1108 DOI: 10.1002/adsc.201000951.

Docekal, V.; Šimek, M.; Dračínský, M.; Vesely, J. Decarboxylative Organocatalytic Allylic Amination of Morita-Baylis-Hillman Carbamates. Chemistry-a European Journal 2018, 24 (51), 13441-13445 DOI: 10.1002/chem.201803677.

Císařová, I.; Docekal, V.; Petrželová, S.; Vesely, J. Enantioselective Cyclopropanation of 4-Nitroisoxazole Derivatives. Advanced Synthesis and Catalysis 2020, 362 (13), 2597-2603 DOI: 10.1002/adsc.202000231.

Vesely, J.; Rios, R. Enantioselective methodologies using N-carbamoyl-imines. Chem. Soc. Rev. 2014, 43 (2), 611-630 DOI: 10.1039/C3CS60321K.

Šimek, M.; Remeš, M.; Vesely, J.; Rios, R. Enantioselective Organocatalytic Amination of Pyrazolones. Asian Journal of Organic Chemistry 2013, 2 (1), 64-68 DOI: 10.1002/ajoc.201200168.

Géant, P. - Y.; Urban, M.; Remeš, M.; Císařová, I.; Vesely, J. Enantioselective Organocatalytic Synthesis of Sulfur-Containing Spirocyclic Compounds: Organocatalytic Synthesis of Sulfur-Containing Spiro Compounds. European Journal of Organic Chemistry 2013, 2013 (35), 7979-7988 DOI: 10.1002/ejoc.201300931.

Zhang, K.; Meazza, M.; Docekal, V.; Light, M. E.; Vesely, J.; Rios, R. Highly Diastereo- and Enantioselective Synthesis of alpha-Spiro-delta-lactams by an Organocascade Reaction. European Journal of Organic Chemistry 2017, No. 13, 1749-1756 DOI: 10.1002/ejoc.201700193.

Kamlar, M.; Bravo, N.; Alba, A. - N. R.; Hybelbauerová, S.; Císařová, I.; Vesely, J.; Moyano, A.; Rios, R. Highly Enantioselective Addition of 1-Fluoro-1-nitro(phenylsulfonyl)methane to α,β-Unsaturated Aldehydes. European Journal of Organic Chemistry 2010, 2010 (28), 5464-5470 DOI: 10.1002/ejoc.201000851.

Franc, M.; Urban, M.; Císařová, I.; Vesely, J. Highly enantioselective addition of sulfur-containing heterocycles to isatin-derived ketimines. Organic & Biomolecular Chemistry 2019, 17 (31), 7309-7314 DOI: 10.1039/c9ob01338e.

Companyó, X.; Hejnová, M.; Kamlar, M.; Vesely, J.; Moyano, A.; Rios, R. Highly enantioselective fluoromalonate addition to α,β-unsaturated aldehydes. Tetrahedron Letters 2009, 50 (35), 5021-5024 DOI: 10.1016/j.tetlet.2009.06.092.

Číhalová, S.; Valero, G.; Schimer, J.; Humpl, M.; Dračínský, M.; Moyano, A.; Rios, R.; Vesely, J. Highly enantioselective organocatalytic cascade reaction for the synthesis of piperidines and oxazolidines. Tetrahedron 2011, 67 (46), 8942-8950 DOI: 10.1016/j.tet.2011.08.079.

Remeš, M.; Vesely, J. Highly Enantioselective Organocatalytic Formation of Functionalized Cyclopentane Derivatives via Tandem Conjugate Addition/α-Alkylation of Enals. European Journal of Organic Chemistry 2012, 2012 (20), 3747-3752 DOI: 10.1002/ejoc.201200334.

Valero, G.; Schimer, J.; Císařová, I.; Vesely, J.; Moyano, A.; Rios, R. Highly enantioselective organocatalytic synthesis of piperidines. Formal synthesis of (−)-Paroxetine. Tetrahedron Letters 2009, 50 (17), 1943-1946 DOI: 10.1016/j.tetlet.2009.02.049.

Kamlar, M.; Vesely, J. Highly enantioselective organocatalytic α-selenylation of aldehydes using hypervalent iodine compounds. Tetrahedron: Asymmetry 2013, 24 (5-6), 254-259 DOI: 10.1016/j.tetasy.2013.02.008.

Vesely, J.; Ledvina, M.; Jindřich, J.; Šaman, D.; Trnka, T. Improved Synthesis of 1,2-trans-Acetates and 1,2-trans Ethyl 1-Thioglycosides Derived from 3,4,6-Tri-O-acetyl-2-deoxy-2-phthalimido-D-hexopyranosides. Collection of Czechoslovak Chemical Communications 2003, 68 (7), 1264-1274 DOI: 10.1135/cccc20031264.

Fanfrlík, J.; Kolář, M.; Kamlar, M.; Hurný, D.; Ruiz, F. X.; Cousido-Siah, A.; Mitschler, A.; Řezáč, J.; Munusamy, E.; Lepšík, M.; et al. Modulation of Aldose Reductase Inhibition by Halogen Bond Tuning. ACS Chemical Biology 2013, 8 (11), 2484-2492 DOI: 10.1021/cb400526n.

Putaj, P.; Tichá, I.; Císařová, I.; Vesely, J. One-Pot Preparation of Chiral Carbacycles from Morita-Baylis-Hillman Carbonates by an Asymmetric Allylic Alkylation/Olefin Metathesis Sequence: One-Pot Preparation of Chiral Carbacycles. European Journal of Organic Chemistry 2014, 2014 (30), 6615-6620 DOI: 10.1002/ejoc.201402899.

Kamlar, M.; Putaj, P.; Vesely, J. Organocatalytic alkynylation of densely functionalized monofluorinated derivatives: C(sp3)–C(sp) coupling. Tetrahedron Letters 2013, 54 (16), 2097-2100 DOI: 10.1016/j.tetlet.2013.02.023.

Vesely, J.; Rios, R. Organocatalytic Enantioselective α-Alkylation of Aldehydes. ChemCatChem 2012, 4 (7), 942-953 DOI: 10.1002/cctc.201200072.

Tsybizova, A.; Remeš, M.; Vesely, J.; Hybelbauerová, S.; Roithová, J. Organocatalytic Preparation of Substituted Cyclopentanes: A Mechanistic Study. The Journal of Organic Chemistry 2014, 79 (4), 1563-1570 DOI: 10.1021/jo4022106.

Humpl, M.; Tauchman, J.; Topolovčan, N.; Kretschmer, J.; Hessler, F.; Císařová, I.; Kotora, M.; Vesely, J. Stereoselective Synthesis of Ezetimibe via Cross-Metathesis of Homoallylalcohols and α-Methylidene-β-Lactams. The Journal of Organic Chemistry 2016, 81 (17), 7692-7699 DOI: 10.1021/acs.joc.6b01406.

Schimer, J.; Cígler, P.; Vesely, J.; Šašková, K. Grantz; Lepšík, M.; Brynda, J.; Řezáčová, P.; Kožíšek, M.; Císařová, I.; Oberwinkler, H.; et al. Structure-Aided Design of Novel Inhibitors of HIV Protease Based on a Benzodiazepine Scaffold. Journal of Medicinal Chemistry 2012, 55 (22), 10130-10135 DOI: 10.1021/jm301249q.

Ceban, V.; Putaj, P.; Meazza, M.; Pitak, M. B.; Coles, S. J.; Vesely, J.; Rios, R. Synergistic catalysis: highly diastereoselective benzoxazole addition to Morita–Baylis–Hillman carbonates. Chemical Communications 2014, 50 (56), 7447 DOI: 10.1039/c4cc00728j.