Publications

Found 163 results
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2020
Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.
Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.
Bultel-Ponce, V.; Durand, T.; Galano, J. - M.; Guy, A.; Jahn, U.; Oger, C.; Pavlíčková, T.; Reversat, G.; Rocher, A.; Vigor, C. First Total Syntheses of Novel Non-Enzymatic Polyunsaturated Fatty Acid Metabolites and Their Identification in Edible Oils. Chemistry - A European Journal 2020, 26 (44), 10090-10098 DOI: 10.1002/chem.202002138.
Bušek, P.; Konvalinka, J.; Šedo, A.; Šimková, A. Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications. Biochimica et Biophysica Acta - Proteins and Proteomics 2020, 1868 (7), nestránkováno DOI: 10.1016/j.bbapap.2020.140409.
Barek, J.; Klouda, J.; Kočovský, P.; Nesměrák, K.; Schwarzova-Peckova, K. A novel voltammetric approach to the detection of primary bile acids in serum samples. Bioelectrochemistry 2020, 134 (August), nestránkováno DOI: 10.1016/j.bioelechem.2020.107539.
Brown, T.; El-Sagheer, A. H.; Hocek, M.; Kellett, A.; Panattoni, A. Oxidative DNA Cleavage with Clip-Phenanthroline Triplex-Forming Oligonucleotide Hybrids. Chembiochem : a European journal of chemical biology 2020, 21 (7), 991-1000 DOI: 10.1002/cbic.201900670.
Beier, P.; Klimánková, I.; Košťál, V.; Motornov, V.; Tichy, D. Preparation of 1-Azido-2-Bromo-1,1,2,2-Tetrafluoroethane and Its Use in the Synthesis of N-Fluoroalkylated Nitrogen Heterocycles. Journal of Organic Chemistry 2020, 85 (17), 11482-11489 DOI: 10.1021/acs.joc.0c01610.
Bastien, G.; Císařová, I.; Dračínský, M.; Hurtado, C. Santos; Kaleta, J.; Mašát, M.; Rogers, C. T.; Rončević, I.; Štoček, J. Radek. Regular Two-Dimensional Arrays of Surface-Mounted Molecular Switches: Switching Monitored by UV-vis and NMR Spectroscopy. Journal of the American Chemical Society 2020, 142 (20), 9337-9351 DOI: 10.1021/jacs.0c01753.
Bursová, M.; Čabala, R.; Hložek, T.; Jelinek, I.; Štícha, M.; Tůma, P. Sensitive CE-MS method for monitoring of riociguat and desmethylriociguat levels in human serum. Electrophoresis 2020, 41 (18-19), 1564-1567 DOI: 10.1002/elps.202000135.
Baszczynski, O.; Cigáň, M.; Filo, J.; Prochazkova, E. Sterically-Controlled Self-Immolation in Phosphoramidate Linkers Triggered by Light. European Journal of Organic Chemistry 2020, 2020 (7), 897-906 DOI: 10.1002/ejoc.201901882.
Brynda, J.; Das, V.; Dvořanová, J.; Džubák, P.; Anwar, S. El; Fábry, M.; Grüner, B.; Gurska, S.; Hajdúch, M.; Havránek, M.; et al. Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX. European Journal of Medicinal Chemistry 2020, 200 (August), nestránkováno DOI: 10.1016/j.ejmech.2020.112460.
Bartova, K.; Džubák, P.; Fleuti, M. Heidi; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Slavětínská, L. Poštová; Tichý, M.; Tloušťová, E. Synthesis and Biological Profiling of Pyrazolo-Fused 7-Deazapurine Nucleosides. Journal of Organic Chemistry 2020, 85 (16), 10539-10551 DOI: 10.1021/acs.joc.0c00928.
Bakhanovich, O.; Beier, P. Synthesis, Stability and Reactivity of alpha-Fluorinated Azidoalkanes. Chemistry - A European Journal 2020, 26 (4), 773-782 DOI: 10.1002/chem.201903627.
Bakhanovich, O.; Beier, P. Synthesis, Stability and Reactivity of alpha-Fluorinated Azidoalkanes. Chemistry - A European Journal 2020, 26 (4), 773-782 DOI: 10.1002/chem.201903627.
Albiñana, C. Berenguer; Brynda, J.; Fanfrlík, J.; Flieger, M.; Hodek, J.; Karlukova, E.; Konvalinka, J.; Kožíšek, M.; Machara, A.; Majer, P.; et al. Unraveling the anti-influenza effect of flavonoids: Experimental validation of luteolin and its congeners as potent influenza endonuclease inhibitors. European Journal of Medicinal Chemistry 2020, 208 (December), nestránkováno DOI: 10.1016/j.ejmech.2020.112754.
2021
Benýšek, J.; Krečmerová, M.; Matoušová, M.; Kaiserová, H. Mertlíkov; Otmar, M.; Pohl, R.; Pomeisl, K.; Pomeislová, A.; Slavětínská, L. Poštová; Rubešová, P. 1,2,4-Thiadiazole acyclic nucleoside phosphonates as inhibitors of cysteine dependent enzymes cathepsin K and GSK-3β. Bioorganic & Medicinal Chemistry 2021, 32 (February), nestránkováno.
Břehová, P.; Česnek, M.; Dračínský, M.; Chaloupecká, E.; Janeba, Z.; Mertlíková-Kaiserová, H.; Skácel, J.; Soto-Velasquez, M. P.; Tloušťová, E.; Watts, V. J. Acyclic nucleoside phosphonates with 2-aminothiazole base as inhibitors of bacterial and mammalian adenylate cyclases. European Journal of Medicinal Chemistry 2021, 222 (October 15 2021), nestránkováno.
Bouřa, E.; Čížek, K.; Eyer, L.; Hocek, M.; Hodek, J.; Konkoľová, E.; Kozák, J.; Milisavljević, N.; Nencka, R.; Pohl, R.; et al. Antiviral Activity of 7-Substituted 7-Deazapurine Ribonucleosides, Monophosphate Prodrugs, and Triphoshates against Emerging RNA Viruses. ACS Infectious Diseases 2021, 7 (2), 471-478.
Bricout, H.; Caronia, E.; Galia, A.; Tichá, I. Chena; Jindřich, J.; Léger, B.; Menuel, S.; Monflier, É.; Noël, S.; Ponchel, A.; et al. Asymmetric hydrogenation of ethyl pyruvate over aqueous dispersed Pt nanoparticles stabilized by a cinchonidine-functionalized β-cyclodextrin. Catalysis Communications 2021, 150 (February), nestránkováno.
Beytlerová, N.; Mateus, M. Alexandre; Kotora, M.; Rýček, L. Catalytic Cyclotrimerization Pathway for Synthesis of Selaginpulvilins C and D: Scope and Limitations. Organic Letters 2021, 23 (12), 4511-4515.
Bělinová, T.; Beneš, H.; Groborz, O.; Heizer, T.; Herynek, V.; Hrubý, M.; Loukotová, L.; Raabová, H.; Švec, P. Direct Comparison of Analogous Amphiphilic Gradient and Block Polyoxazolines. Macromolecules 2021, 54 (17), 8182-8194.
Bělinová, T.; Beneš, H.; Groborz, O.; Heizer, T.; Herynek, V.; Hrubý, M.; Loukotová, L.; Raabová, H.; Švec, P. Direct Comparison of Analogous Amphiphilic Gradient and Block Polyoxazolines. Macromolecules 2021, 54 (17), 8182-8194.
Baszczyňski, O.; Dračínský, M.; Dvořáková, A.; Hodek, J.; Chalupský, K.; Janeba, Z.; Kalčic, F.; Kaiserová, H. Mertlíkov; Strmeň, T.; Šebestík, J.; et al. Discovery of Modified Amidate (ProTide) Prodrugs of Tenofovir with Enhanced Antiviral Properties. Journal of Medicinal Chemistry 2021, 64 (22), 16425-16449.
Beier, P.; Chvojka, T.; Janecký, L.; Klepetářová, B.; Markos, A.; Martínek, T.; Martinez-Seara, H. Haloalkenyl Imidoyl Halides as Multifacial Substrates in the Stereoselective Synthesis of N-Alkenyl Compounds. Advanced Synthesis and Catalysis 2021, 363 (13), 3258-3266.
Bednářová, E.; Kotora, M.; Malatinec, Š.; Tanaka, H. Highly Enantioselective Ring-Opening of meso-Epoxides with O- and N-Nucleophiles Catalyzed by a Chiral Sc(III)/bipyridine Complex. European Journal of Organic Chemistry 2021, 2021 (8), 1249-1257.
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