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Found 140 results
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2023
Štefek, M.; Chalupská, D.; Chalupský, K.; Zgarbová, M.; Dvořáková, A.; Krafčíková, P.; Li, A. Shi Ming; Šála, M.; Dejmek, M.; Otava, T.; et al. Rational Design of Highly Potent SARS-CoV-2 nsp14 Methyltransferase Inhibitors. ACS Omega 2023, 8 (30), 27410-27418.
Lončarić, D.; Movahedifar, F.; Štoček, J. Radek; Dračínský, M.; Cvačka, J.; Guan, S.; Bythell, B. J.; Císařová, I.; Masson, E.; Kaleta, J. Solvent-controlled formation of alkali and alkali-earth-secured cucurbituril/guest trimers. Chemical Science 2023, 14 (35), 9258-9266.
Lóška, L.; Dočekal, V.; Císařová, I.; Veselý, J. Stereoselective N-Heterocyclic-Carbene-Catalyzed Formal [4+2] Cycloaddition: Access to Chiral Heterocyclic Cyclohexenones. Organic Letters 2023, 25 (1), 174-178.
Yang, C.; Tichý, M.; Slavětínská, L. Poštová; Vaiedelich, E.; Gurská, S.; Džubák, P.; Hajdúch, M.; Hocek, M. Synthesis and Biological Profiling of Benzofuro-Fused 7-Deazapurine Nucleosides. European Journal of Organic Chemistry 2023, 26 (44).
Lapinskaite, R.; Atalay, H. Nazlican; Malatinec, Š.; Dönmez, S.; Cinar, Z. Özlem; Schwarz, P. F.; Perhal, A. F.; Císařová, I.; Labanauskas, L.; Karpiński, T. M.; et al. Synthesis of Selagibenzophenone A and Its Derivatives for Evaluation of Their Antiproliferative, ROR gamma Inverse Agonistic, and Antimicrobial Effect. ChemistrySelect 2023, 8 (7).
Lapinskaite, R.; Atalay, H. Nazlican; Malatinec, Š.; Dönmez, S.; Cinar, Z. Özlem; Schwarz, P. F.; Perhal, A. F.; Císařová, I.; Labanauskas, L.; Karpiński, T. M.; et al. Synthesis of Selagibenzophenone A and Its Derivatives for Evaluation of Their Antiproliferative, ROR gamma Inverse Agonistic, and Antimicrobial Effect. ChemistrySelect 2023, 8 (7).
Dejmek, M.; Brázdová, A.; Otava, T.; Polidarová, M. Pimková; Klíma, M.; Smola, M.; Vavřina, Z.; Buděšínský, M.; Dračínský, M.; Liboska, R.; et al. Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy. European Journal of Medicinal Chemistry 2023, 259 (November).
Dejmek, M.; Brázdová, A.; Otava, T.; Polidarová, M. Pimková; Klíma, M.; Smola, M.; Vavřina, Z.; Buděšínský, M.; Dračínský, M.; Liboska, R.; et al. Vinylphosphonate-based cyclic dinucleotides enhance STING-mediated cancer immunotherapy. European Journal of Medicinal Chemistry 2023, 259 (November).
Díaz-Holguín, A.; Rashidian, A.; Pijnenburg, D.; Ferreira, G. Monteiro; Štefela, A.; Kašpar, M.; Kudová, E.; Poso, A.; van Beuningen, R.; Pávek, P.; et al. When Two Become One: Conformational Changes in FXR/RXR Heterodimers Bound to Steroidal Antagonists. ChemMedChem 2023, 18 (4).
2022
Čikoš, A.; Degač, M.; Gredičak, M.; Topolovčan, N. Chemoselective and Regioselective Synthesis of Spiroisoindolinone Indenes via an Intercepted Meyer–Schuster Rearrangement/Intramolecular Friedel–Crafts Alkylation Relay. Journal of Organic Chemistry 2022, 87 (5), 3712-3717.
Dian, J.; Fourmentin, S.; Jindřich, J.; Palágyi, A. Cyclodextrin-based Schiff base pro-fragrances: Synthesis and release studies. Beilstein Journal of Organic Chemistry 2022, 18 (September), 1346-1354.
Ausserlechner, M. J.; Dočekal, V.; Hagenbuchner, J.; Horváth, M.; Kaiser, N.; Kohoutová, K.; Mandal, R.; Obšil, T.; Obšilová, V.; Tekel, A.; et al. Lengthening the Guanidine–Aryl Linker of Phenylpyrimidinylguanidines Increases Their Potency as Inhibitors of FOXO3-Induced Gene Transcription. ACS Omega [online] 2022, 7 (38), 34632-34646.
Ausserlechner, M.; Dočekal, V.; Kohoutová, K.; Obšil, T.; Obšilová, V.; Tekel, A.; Veselý, J. Modulating FOXO3 transcriptional activity by low-molecular compounds. FEBS Open Bio [online], 2022, 12, 233-233.
Císařová, I.; David, T.; Dračínský, M.; Jirák, D.; Jurok, R.; Kretschmer, J.; Kuchař, M.; Polášek, M.; Socha, O.; Vít, M. Paramagnetic encoding of molecules. Nature Communications [online] 2022, 13 (1), nestránkováno.
Císařová, I.; David, T.; Dračínský, M.; Jirák, D.; Jurok, R.; Kretschmer, J.; Kuchař, M.; Polášek, M.; Socha, O.; Vít, M. Paramagnetic encoding of molecules. Nature Communications [online] 2022, 13 (1), nestránkováno.
Císařová, I.; Dočekal, V.; Gyepes, R.; Hrabovský, J.; Koberová, T.; Rios, R.; Veselý, J.; Vopálenská, A. Stereoselective cyclopropanation of boron dipyrromethene (BODIPY) derivatives by an organocascade reaction. Advanced Synthesis and Catalysis 2022, 364 (5), 930-937.
Bouřa, E.; Dejmek, M.; Chalupská, D.; Klíma, M.; Matoušová, M.; Mertlíková-Kaiserová, H.; Misehe, M.; Nencka, R.; Šála, M. Structure-based design and modular synthesis of novel PI4K class II inhibitors bearing a 4-aminoquinazoline scaffold. Bioorganic and Medicinal Chemistry Letters 2022, 76 (November), nestránkováno.
2021
Břehová, P.; Česnek, M.; Dračínský, M.; Chaloupecká, E.; Janeba, Z.; Mertlíková-Kaiserová, H.; Skácel, J.; Soto-Velasquez, M. P.; Tloušťová, E.; Watts, V. J. Acyclic nucleoside phosphonates with 2-aminothiazole base as inhibitors of bacterial and mammalian adenylate cyclases. European Journal of Medicinal Chemistry 2021, 222 (October 15 2021), nestránkováno.
Baszczyňski, O.; Dračínský, M.; Dvořáková, A.; Hodek, J.; Chalupský, K.; Janeba, Z.; Kalčic, F.; Kaiserová, H. Mertlíkov; Strmeň, T.; Šebestík, J.; et al. Discovery of Modified Amidate (ProTide) Prodrugs of Tenofovir with Enhanced Antiviral Properties. Journal of Medicinal Chemistry 2021, 64 (22), 16425-16449.
Baszczyňski, O.; Dračínský, M.; Dvořáková, A.; Hodek, J.; Chalupský, K.; Janeba, Z.; Kalčic, F.; Kaiserová, H. Mertlíkov; Strmeň, T.; Šebestík, J.; et al. Discovery of Modified Amidate (ProTide) Prodrugs of Tenofovir with Enhanced Antiviral Properties. Journal of Medicinal Chemistry 2021, 64 (22), 16425-16449.
Dračínský, M.; Drastík, M.; Kašpar, M.; Klepetářová, B.; Kronenberger, T.; Kudová, E.; Mičuda, S.; Pávek, P.; Štefela, A. (E)-7-Ethylidene-lithocholic Acid (7-ELCA) Is a Potent Dual Farnesoid X Receptor (FXR) Antagonist and GPBAR1 Agonist Inhibiting FXR-Induced Gene Expression in Hepatocytes and Stimulating Glucagon-like Peptide-1 Secretion From Enteroendocrine Cells. Frontiers in Pharmacology 2021, 12 (August), nestránkováno.
Dračínský, M.; Drastík, M.; Kašpar, M.; Klepetářová, B.; Kronenberger, T.; Kudová, E.; Mičuda, S.; Pávek, P.; Štefela, A. (E)-7-Ethylidene-lithocholic Acid (7-ELCA) Is a Potent Dual Farnesoid X Receptor (FXR) Antagonist and GPBAR1 Agonist Inhibiting FXR-Induced Gene Expression in Hepatocytes and Stimulating Glucagon-like Peptide-1 Secretion From Enteroendocrine Cells. Frontiers in Pharmacology 2021, 12 (August), nestránkováno.
Doleželová, E.; Downey, A. Michael; Hocek, M.; Nguyen, V. Hai; Pohl, R.; Rožánková, S.; Slapničková, M.; Tichý, M.; Tloušťová, E.; Zíková, A. Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides. Bioorganic and Medicinal Chemistry Letters 2021, 40 (May 15 2021), nestránkováno.
Doleželová, E.; Downey, A. Michael; Hocek, M.; Nguyen, V. Hai; Pohl, R.; Rožánková, S.; Slapničková, M.; Tichý, M.; Tloušťová, E.; Zíková, A. Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides. Bioorganic and Medicinal Chemistry Letters 2021, 40 (May 15 2021), nestránkováno.
Doleželová, E.; Džubák, P.; Gurská, S.; Hajdúch, M.; Hocek, M.; Krajczyk, A.; Milisavljević, N.; Perlíková, P.; Slavětínská, L. Poštová; Slapničková, M.; et al. Synthesis and Antitrypanosomal Activity of 6-Substituted 7-Methyl-7-deazapurine Nucleosides. ACS Infectious Diseases 2021, 7 (4), 917-926.
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