Publications

Found 502 results
Author Title Type [ Year(Desc)]
2023
Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.
Novotná, K.; Tenora, L.; Prchalová, E.; Paule, J.; Alt, J.; Veeravalli, V.; Lam, J.; Wu, Y.; Šnajdr, I.; Gori, S.; et al. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry 2023, 66 (22), 15493-15510.
Holovko-Kamoshenkova, O. M.; Slivka, M. V.; Hrdina, R.; Baumer, V. N.; Korol, N. I.; Sokolenko, L. V.; Lendel, V. G. An Efficient Catalyst-Free Direct Approach to 5-Polyfluoroalkyl-1,2,4-triazole-3-thiones. Synthesis 2023, 55 (08), 1221-1226.
Spampinato, A.; Kužmová, E.; Pohl, R.; Sýkorová, V.; Vrábel, M.; Kraus, T.; Hocek, M. trans-Cyclooctene- and Bicyclononyne-Linked Nucleotides for Click Modification of DNA with Fluorogenic Tetrazines and Live Cell Metabolic Labeling and Imaging. Bioconjugate Chemistry 2023, 34 (4), 772-780.
Belhajová, M.; Vícha, A.; Burgert, L.; Brožková, I.; Michaličková, L.; Hrdina, R.; Moravec, T.; Netuka, D.; Musil, Z.; Hrdina, R. En route to local glioblastoma treatment with temozolomide doped hyaluronan fibres: formulation and in vitro cell studies. RSC Medicinal Chemistry 2023, 14 (9), 1662-1666.
Nigríni, M.; Bhosale, V. Anandrao; Císařová, I.; Veselý, J. Enantioenriched 1,4-Benzoxazepines via Chiral Brønsted Acid-Catalyzed Enantioselective Desymmetrization of 3-Substituted Oxetanes. Journal of Organic Chemistry 2023, 88 (24), 17024-17036.
Kamlar, M.; Urban, M.; Veselý, J. Enantioselective Synthesis of Spiro Heterocyclic Compounds Using a Combination of Organocatalysis and Transition-Metal Catalysis. Chemical Record 2023, 23 (7).
Misehe, M.; Matoušová, M.; Dvořáková, A.; Hercík, K.; Škach, K.; Chalupská, D.; Dejmek, M.; Šála, M.; Hájek, M.; Bouřa, E.; et al. Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases. European Journal of Medicinal Chemistry 2023, 260 (November).
Ortiz, M.; Jauset-Rubio, M.; Trummer, O.; Foessl, I.; Kodr, D.; Acero, J. Lluís; Botero, M. Luz; Biggs, P.; Lenartowicz, D.; Trajanoska, K.; et al. Generic Platform for the Multiplexed Targeted Electrochemical Detection of Osteoporosis-Associated Single Nucleotide Polymorphisms Using Recombinase Polymerase Solid-Phase Primer Elongation and Ferrocene-Modified Nucleoside Triphosphates. ACS Central Science 2023, 9 (8), 1591-1602.
Coufal, R.; Tošner, Z.; Drahoňovský, D.; Vohlídal, J. Hemiacetal-based dynamic systems: a new mechanistic insight. Organic and Biomolecular Chemistry 2023, 21 (34), 6956-6968.
Osifová, Z.; Šála, M.; Dračínský, M. Hydrogen-Bonding Interactions of 8-Substituted Purine Derivatives. ACS Omega 2023, 8 (28), 25538-25548.
Kugler, M.; Hadzima, M.; Dzijak, R.; Rampmaier, R.; Srb, P.; Vrzal, L.; Voburka, Z.; Majer, P.; Řezáčová, P.; Vrábel, M. Identification of specific carbonic anhydrase inhibitors via in situ click chemistry, phage-display and synthetic peptide libraries: comparison of the methods and structural study. RSC Medicinal Chemistry 2023, 14 (1), 144-153.
Janecký, L.; Markos, A.; Klepetářová, B.; Beier, P. Lewis-Acid-Mediated Intramolecular Cyclization of 4-Aryl-5-allyl-1,2,3-triazoles to Substituted Cyclopentene Derivatives. Journal of Organic Chemistry 2023, 88 (2), 1155-1167.
Kodr, D.; Kužmová, E.; Pohl, R.; Kraus, T.; Hocek, M. Lipid-linked nucleoside triphosphates for enzymatic synthesis of hydrophobic oligonucleotides with enhanced membrane anchoring efficiency. Chemical Science 2023, 14 (15), 4059-4069.
Navrátil, R.; Kellovská, K.; Baszczyňski, O. Multimetallic Pd- and Ni-catalyzed C(sp2)–P cross-coupling under aqueous micellar conditions. Green Chemistry 2023, 25 (23), 9779-9794.
Novotná, K.; Thomas, A. G.; Štěpánek, O.; Murphy, B.; Hin, N.; Skácel, J.; Mueller, L.; Tenora, L.; Pal, A.; Alt, J.; et al. Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a] scaffold. European Journal of Medicinal Chemistry 2023, 259 (November).
Socha, O.; Osifová, Z.; Dračínský, M. NMR-Challenge.com: An Interactive Website with Exercises in Solving Structures from NMR Spectra. Journal of Chemical Education 2023, 100 (2), 962-968.
Kodr, D.; Ortiz, M.; Sýkorová, V.; Yenice, C. Pinar; Lesnikowski, Z. J.; O’Sullivan, C. K.; Hocek, M. Normalized Multipotential Redox Coding of DNA Bases for Determination of Total Nucleotide Composition. Analytical Chemistry 2023, 95 (34), 12586-12589.
Kuba, M.; Pohl, R.; Kraus, T.; Hocek, M. Nucleotides Bearing Red Viscosity-Sensitive Dimethoxy-Bodipy Fluorophore for Enzymatic Incorporation and DNA Labeling. Bioconjugate Chemistry 2023, 34 (1), 133-139.
Kamlar, M.; Císařová, I.; Veselý, J. PCCP-Catalyzed Synthesis of Tetrasubstituted Allenes Bearing Heteroaromatic Sulfenyl Group. European Journal of Organic Chemistry 2023, 26 (32).
Runemark, A.; Martos, M.; Nigríni, M.; Noa, F. M. Amombo; Öhrström, L.; Sunden, H. Photochemical Access to Substituted β-Lactams and β-Lactones via the Zimmerman–O’Connell–Griffin Rearrangement. Organic Letters 2023, 25 (29), 5520-5524.
Lebedinskiy, K.; Jindřich, J. Preparation of 6-Monohalo-β-cyclodextrin Derivatives with Selectively Methylated Rims via Diazonium Salts. ACS Omega 2023, 8 (31), 28268-28276.
Kurbanova, A.; Nigríni, M.; Gołąbek, K. Maria; Veselý, O.; Veselý, J. Preparation of functionalised tetrahydropyrans catalysed by isoreticular zeolites. Microporous and Mesoporous Materials 2023, 350 (February).
Štefek, M.; Chalupská, D.; Chalupský, K.; Zgarbová, M.; Dvořáková, A.; Krafčíková, P.; Li, A. Shi Ming; Šála, M.; Dejmek, M.; Otava, T.; et al. Rational Design of Highly Potent SARS-CoV-2 nsp14 Methyltransferase Inhibitors. ACS Omega 2023, 8 (30), 27410-27418.
Kuba, M.; Khoroshyy, P.; Lepšík, M.; Kužmová, E.; Kodr, D.; Kraus, T.; Hocek, M. Real-time Imaging of Nascent DNA in Live Cells by Monitoring the Fluorescence Lifetime of DNA-Incorporated Thiazole Orange-Modified Nucleotides. Angewandte Chemie - International Edition 2023, 62 (38).
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