Publications

Brynda, J.; Fanfrlík, J.; Hadzima, M.; Hánová, I.; Horn, M.; Houštecká, R.; Lepšík, M.; Majer, P.; Mareš, M.; Mertlíková-Kaiserová, H.; et al. Biomimetic Macrocyclic Inhibitors of Human Cathepsin D: Structure-Activity Relationship and Binding Mode Analysis. Journal of Medicinal Chemistry 2020, 63 (4), 1576-1596 DOI: 10.1021/acs.jmedchem.9b01351.

Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.

Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.

Bultel-Ponce, V.; Durand, T.; Galano, J. - M.; Guy, A.; Jahn, U.; Oger, C.; Pavlíčková, T.; Reversat, G.; Rocher, A.; Vigor, C. First Total Syntheses of Novel Non-Enzymatic Polyunsaturated Fatty Acid Metabolites and Their Identification in Edible Oils. Chemistry - A European Journal 2020, 26 (44), 10090-10098 DOI: 10.1002/chem.202002138.

Bušek, P.; Konvalinka, J.; Šedo, A.; Šimková, A. Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications. Biochimica et Biophysica Acta - Proteins and Proteomics 2020, 1868 (7), nestránkováno DOI: 10.1016/j.bbapap.2020.140409.

Barek, J.; Klouda, J.; Kočovský, P.; Nesměrák, K.; Schwarzova-Peckova, K. A novel voltammetric approach to the detection of primary bile acids in serum samples. Bioelectrochemistry 2020, 134 (August), nestránkováno DOI: 10.1016/j.bioelechem.2020.107539.

Brown, T.; El-Sagheer, A. H.; Hocek, M.; Kellett, A.; Panattoni, A. Oxidative DNA Cleavage with Clip-Phenanthroline Triplex-Forming Oligonucleotide Hybrids. Chembiochem : a European journal of chemical biology 2020, 21 (7), 991-1000 DOI: 10.1002/cbic.201900670.

Beier, P.; Klimánková, I.; Košťál, V.; Motornov, V.; Tichy, D. Preparation of 1-Azido-2-Bromo-1,1,2,2-Tetrafluoroethane and Its Use in the Synthesis of N-Fluoroalkylated Nitrogen Heterocycles. Journal of Organic Chemistry 2020, 85 (17), 11482-11489 DOI: 10.1021/acs.joc.0c01610.

Bastien, G.; Císařová, I.; Dračínský, M.; Hurtado, C. Santos; Kaleta, J.; Mašát, M.; Rogers, C. T.; Rončević, I.; Štoček, J. Radek. Regular Two-Dimensional Arrays of Surface-Mounted Molecular Switches: Switching Monitored by UV-vis and NMR Spectroscopy. Journal of the American Chemical Society 2020, 142 (20), 9337-9351 DOI: 10.1021/jacs.0c01753.

Bursová, M.; Čabala, R.; Hložek, T.; Jelinek, I.; Štícha, M.; Tůma, P. Sensitive CE-MS method for monitoring of riociguat and desmethylriociguat levels in human serum. Electrophoresis 2020, 41 (18-19), 1564-1567 DOI: 10.1002/elps.202000135.

Baszczynski, O.; Cigáň, M.; Filo, J.; Prochazkova, E. Sterically-Controlled Self-Immolation in Phosphoramidate Linkers Triggered by Light. European Journal of Organic Chemistry 2020, 2020 (7), 897-906 DOI: 10.1002/ejoc.201901882.

Brynda, J.; Das, V.; Dvořanová, J.; Džubák, P.; Anwar, S. El; Fábry, M.; Grüner, B.; Gurska, S.; Hajdúch, M.; Havránek, M.; et al. Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX. European Journal of Medicinal Chemistry 2020, 200 (August), nestránkováno DOI: 10.1016/j.ejmech.2020.112460.

Bartova, K.; Džubák, P.; Fleuti, M. Heidi; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Slavětínská, L. Poštová; Tichý, M.; Tloušťová, E. Synthesis and Biological Profiling of Pyrazolo-Fused 7-Deazapurine Nucleosides. Journal of Organic Chemistry 2020, 85 (16), 10539-10551 DOI: 10.1021/acs.joc.0c00928.

Bakhanovich, O.; Beier, P. Synthesis, Stability and Reactivity of alpha-Fluorinated Azidoalkanes. Chemistry - A European Journal 2020, 26 (4), 773-782 DOI: 10.1002/chem.201903627.

Bakhanovich, O.; Beier, P. Synthesis, Stability and Reactivity of alpha-Fluorinated Azidoalkanes. Chemistry - A European Journal 2020, 26 (4), 773-782 DOI: 10.1002/chem.201903627.

Albiñana, C. Berenguer; Brynda, J.; Fanfrlík, J.; Flieger, M.; Hodek, J.; Karlukova, E.; Konvalinka, J.; Kožíšek, M.; Machara, A.; Majer, P.; et al. Unraveling the anti-influenza effect of flavonoids: Experimental validation of luteolin and its congeners as potent influenza endonuclease inhibitors. European Journal of Medicinal Chemistry 2020, 208 (December), nestránkováno DOI: 10.1016/j.ejmech.2020.112754.

Prochazkova, E.; Navrátil, R.; Janeba, Z.; Roithová, J.; Baszczynski, O. Reactive cyclic intermediates in the ProTide prodrugs activation: trapping the elusive pentavalent phosphorane. Organic & Biomolecular Chemistry 2019, 17 (2), 315-320 DOI: 10.1039/c8ob02870b.

Kulkarni, R.; Noda, Y.; Barange, D. Kumar; Kochergin, Y. S.; Lyu, P.; Balcarova, B.; Nachtigall, P.; Bojdys, M. J. Real-time optical and electronic sensing with a beta-amino enone linked, triazine-containing 2D covalent organic framework. Nature Communications 2019, 10, 3228 DOI: 10.1038/s41467-019-11264-z.

Kulkarni, R.; Noda, Y.; Barange, D. Kumar; Kochergin, Y. S.; Lyu, P.; Balcarova, B.; Nachtigall, P.; Bojdys, M. J. Real-time optical and electronic sensing with a beta-amino enone linked, triazine-containing 2D covalent organic framework. Nature Communications 2019, 10, 3228 DOI: 10.1038/s41467-019-11264-z.

Kulkarni, R.; Noda, Y.; Barange, D. Kumar; Kochergin, Y. S.; Lyu, P.; Balcarova, B.; Nachtigall, P.; Bojdys, M. J. Real-time optical and electronic sensing with a beta-amino enone linked, triazine-containing 2D covalent organic framework. Nature Communications 2019, 10, 3228 DOI: 10.1038/s41467-019-11264-z.

Markos, A.; Voltrova, S.; Motornov, V.; Tichy, D.; Klepetářová, B.; Beier, P. Stereoselective Synthesis of (Z)-beta-Enamido Triflates and Fluorosulfonates from N-Fluoroalkylated Triazoles. Chemistry-a European Journal 2019, 25 (32), 7640-7644 DOI: 10.1002/chem.201901632.

Bris, A.; Turel, I.; Roithová, J. C-H Bond Activation by a Ruthenium(II) beta-Diketonate Complex: A Mechanistic Study. European Journal of Organic Chemistry 2018, No. 44, 6107-6113 DOI: 10.1002/ejoc.201800787.

Kochergin, Y. S.; Schwarz, D.; Acharjya, A.; Ichangi, A.; Kulkarni, R.; Eliasova, P.; Vacek, J.; Schmidt, J.; Thomas, A.; Bojdys, M. J. Exploring the "Goldilocks Zone" of Semiconducting Polymer Photocatalysts by Donor-Acceptor Interactions. Angewandte Chemie-International Edition 2018, 57 (43), 14188-14192 DOI: 10.1002/anie.201809702.

Schwarz, D.; Acharja, A.; Ichangi, A.; Lyu, P.; Opanasenko, M. V.; Gossler, F. R.; Konig, T. A. F.; Cejka, J.; Nachtigall, P.; Thomas, A.; et al. Fluorescent Sulphur- and Nitrogen-Containing Porous Polymers with Tuneable Donor-Acceptor Domains for Light-Driven Hydrogen Evolution. Chemistry-a European Journal 2018, 24 (46), 11916-11921 DOI: 10.1002/chem.201802902.

Krömer, M.; Bartova, K.; Raindlová, V.; Hocek, M. Synthesis of Dihydroxyalkynyl and Dihydroxyalkyl Nucleotides as Building Blocks or Precursors for Introduction of Diol or Aldehyde Groups to DNA for Bioconjugations. Chemistry-a European Journal 2018, 24 (46), 11890-11894 DOI: 10.1002/chem.201802282.