Publications

Urban, M.; Franc, M.; Hofmanova, M.; Císařová, I.; Veselý, J. The enantioselective addition of 1-fluoro-1-nitro (phenylsulfonyl) methane to isatin-derived ketimines. Organic & Biomolecular Chemistry 2017, 15 (43), 9071-9076 DOI: 10.1039/c7ob02408h.

Kopecna, M.; Machacek, M.; Prchalová, E.; Stepanek, P.; Drasar, P.; Kotora, M.; Vavrova, K. Galactosyl Pentadecene Reversibly Enhances Transdermal and Topical Drug Delivery. Pharmaceutical Research 2017, 34 (10), 2097-2108 DOI: 10.1007/s11095-017-2214-3.

Zhang, K.; Meazza, M.; Docekal, V.; Light, M. E.; Vesely, J.; Rios, R. Highly Diastereo- and Enantioselective Synthesis of alpha-Spiro-delta-lactams by an Organocascade Reaction. European Journal of Organic Chemistry 2017, No. 13, 1749-1756 DOI: 10.1002/ejoc.201700193.

Trautner, S.; Jašík, J.; Parigger, C. G.; Pedarnig, J. D.; Spendelhofer, W.; Lackner, J.; Veis, P.; Heitz, J. Laser-induced optical breakdown spectroscopy of polymer materials based on evaluation of molecular emission bands (vol 174, pg 331, 2017). Spectrochimica Acta Part a-Molecular and Biomolecular Spectroscopy 2017, 179, 73-73 DOI: 10.1016/j.saa.2017.02.016.

Trautner, S.; Jašík, J.; Parigger, C. G.; Pedarnig, J. D.; Spendelhofer, W.; Lackner, J.; Veis, P.; Heitz, J. Laser-induced optical breakdown spectroscopy of polymer materials based on evaluation of molecular emission bands. Spectrochimica Acta Part a-Molecular and Biomolecular Spectroscopy 2017, 174, 331-338 DOI: 10.1016/j.saa.2016.11.045.

Váňa, J.; Lang, J.; Soltesova, M.; Hanusek, J.; Růžička, A.; Sedlák, M.; Roithová, J. The role of trinuclear species in a palladium acetate/trifluoroacetic acid catalytic system. Dalton Transactions 2017, 46 (46), 16269-16275 DOI: 10.1039/c7dt03832a.

Humpl, M.; Tauchman, J.; Topolovčan, N.; Kretschmer, J.; Hessler, F.; Císařová, I.; Kotora, M.; Vesely, J. Stereoselective Synthesis of Ezetimibe via Cross-Metathesis of Homoallylalcohols and α-Methylidene-β-Lactams. The Journal of Organic Chemistry 2016, 81 (17), 7692-7699 DOI: 10.1021/acs.joc.6b01406.

Kamlar, M.; Císařová, I.; Veselý, J. Alkynylation of heterocyclic compounds using hypervalent iodine reagent. Org. Biomol. Chem. 2015, 13 (10), 2884-2889 DOI: 10.1039/C4OB02625J.

Dadová, J.; Vrábel, M.; Adámik, M.; Brázdová, M.; Pohl, R.; Fojta, M.; Hocek, M. Azidopropylvinylsulfonamide as a New Bifunctional Click Reagent for Bioorthogonal Conjugations: Application for DNA-Protein Cross-Linking. Chemistry - A European Journal 2015, 21 (45), 16091-16102 DOI: 10.1002/chem.201502209.

Gergelitsová, I.; Tauchman, J.; Císařová, I.; Veselý, J. Bifunctional (Thio)urea–Phosphine Organocatalysts Derived from d-Glucose and α-Amino Acids and Their Application to the Enantio­selective Morita–Baylis–Hillman Reaction. Synlett 2015, 26 (19), 2690-2696 DOI: 10.1055/s-0035-1560931.

Motloch, P.; Valterová, I.; Kotora, M. Enantioselective Allylation of Thiophene-2-carbaldehyde: Formal Total Synthesis of Duloxetine. Advanced Synthesis & Catalysis 2014, 356 (1), 199-204 DOI: 10.1002/adsc.201300849.

Vesely, J.; Rios, R. Enantioselective methodologies using N-carbamoyl-imines. Chem. Soc. Rev. 2014, 43 (2), 611-630 DOI: 10.1039/C3CS60321K.

Hanzlová, E.; Váňa, J.; Shaffer, C. J.; Roithová, J.; Martinů, T. Evidence for the Cyclic CN ₂ Carbene in the Gas Phase. Organic Letters 2014, 16 (20), 5482-5485 DOI: 10.1021/ol5027602.

Tumova, L.; Pombinho, A. R.; Vojtechova, M.; Stancikova, J.; Gradl, D.; Krausova, M.; Sloncova, E.; Horazna, M.; Kriz, V.; Machonova, O.; et al. Monensin inhibits canonical wnt signaling in human colorectal cancer cells and suppresses tumor growth in multiple intestinal neoplasia mice. Molecular cancer therapeutics 2014, 13 (4), 812-822 DOI: 10.1158/1535-7163.MCT-13-0625.

Putaj, P.; Tichá, I.; Císařová, I.; Vesely, J. One-Pot Preparation of Chiral Carbacycles from Morita-Baylis-Hillman Carbonates by an Asymmetric Allylic Alkylation/Olefin Metathesis Sequence: One-Pot Preparation of Chiral Carbacycles. European Journal of Organic Chemistry 2014, 2014 (30), 6615-6620 DOI: 10.1002/ejoc.201402899.

Kamlar, M.; Hybelbauerová, S.; Císařová, I.; Veselý, J. Organocatalytic enantioselective allylic alkylation of MBH carbonates with β-keto esters. Organic & Biomolecular Chemistry 2014, 12 (28), 5071 DOI: 10.1039/c4ob00682h.

Tsybizova, A.; Remeš, M.; Vesely, J.; Hybelbauerová, S.; Roithová, J. Organocatalytic Preparation of Substituted Cyclopentanes: A Mechanistic Study. The Journal of Organic Chemistry 2014, 79 (4), 1563-1570 DOI: 10.1021/jo4022106.

Vaníková, Z.; Hocek, M. Polymerase Synthesis of Photocaged DNA Resistant against Cleavage by Restriction Endonucleases. Angewandte Chemie International Edition 2014, 53 (26), 6734-6737 DOI: 10.1002/anie.201402370.

Váňa, J.; Roithová, J.; Kotora, M.; Beran, P.; Rulíšek, L.; Kočovský, P. Proton Affinities of Organocatalysts Derived from Pyridine N-oxide. Croatica Chemica Acta 2014, 87 (4), 349-356 DOI: 10.5562/cca2447.

Snášel, J.; Nauš, P.; Dostál, J.; Hnízda, A.; Fanfrlík, J.; Brynda, J.; Bourderioux, A.; Dušek, M.; Dvořáková, H.; Stolaříková, J.; et al. Structural Basis for Inhibition of Mycobacterial and Human Adenosine Kinase by 7-Substituted 7-(Het)aryl-7-deazaadenine Ribonucleosides. Journal of Medicinal Chemistry 2014, 57 (20), 8268-8279 DOI: 10.1021/jm500497v.

Snášel, J.; Nauš, P.; Dostál, J.; Hnízda, A.; Fanfrlík, J.; Brynda, J.; Bourderioux, A.; Dušek, M.; Dvořáková, H.; Stolaříková, J.; et al. Structural Basis for Inhibition of Mycobacterial and Human Adenosine Kinase by 7-Substituted 7-(Het)aryl-7-deazaadenine Ribonucleosides. Journal of Medicinal Chemistry 2014, 57 (20), 8268-8279 DOI: 10.1021/jm500497v.

Ceban, V.; Putaj, P.; Meazza, M.; Pitak, M. B.; Coles, S. J.; Vesely, J.; Rios, R. Synergistic catalysis: highly diastereoselective benzoxazole addition to Morita–Baylis–Hillman carbonates. Chemical Communications 2014, 50 (56), 7447 DOI: 10.1039/c4cc00728j.

Hessler, F.; Korotvička, A.; Nečas, D.; Valterová, I.; Kotora, M. Syntheses of a Flobufen Metabolite and Dapoxetine Based on Enantioselective Allylation of Aromatic Aldehydes: Syntheses of a Flobufen Metabolite and Dapoxetine. European Journal of Organic Chemistry 2014, 2014 (12), 2543-2548 DOI: 10.1002/ejoc.201301899.

Nauš, P.; Caletková, O.; Konečný, P.; Džubák, P.; Bogdanová, K.; Kolář, M.; Vrbková, J.; Slavětínská, L.; Tloušt’ová, E.; Perlíková, P.; et al. Synthesis, Cytostatic, Antimicrobial, and Anti-HCV Activity of 6-Substituted 7-(Het)aryl-7-deazapurine Ribonucleosides. Journal of Medicinal Chemistry 2014, 57 (3), 1097-1110 DOI: 10.1021/jm4018948.

Perlíková, P.; Konečný, P.; Nauš, P.; Snášel, J.; Votruba, I.; Džubák, P.; Pichová, I.; Hajdúch, M.; Hocek, M. 6-Alkyl-, 6-aryl- or 6-hetaryl-7-deazapurine ribonucleosides as inhibitors of human or MTB adenosine kinase and potential antimycobacterial agents. MedChemComm 2013, 4 (11), 1497 DOI: 10.1039/c3md00232b.