Publications

Found 264 results
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2020
Drastík, M.; Holas, O.; Hroch, M.; Hutníková, M.; Kašpar, M.; Kudová, E.; Mičuda, S.; Pandey, A. V.; Pávek, P.; Smutný, T.; et al. 3 beta-Isoobeticholic acid efficiently activates the farnesoid X receptor (FXR) due to its epimerization to 3 alpha-epimer by hepatic metabolism. Journal of Steroid Biochemistry and Molecular Biology 2020, 202 (September), nestránkováno DOI: 10.1016/j.jsbmb.2020.105702.
Drastík, M.; Holas, O.; Hroch, M.; Hutníková, M.; Kašpar, M.; Kudová, E.; Mičuda, S.; Pandey, A. V.; Pávek, P.; Smutný, T.; et al. 3 beta-Isoobeticholic acid efficiently activates the farnesoid X receptor (FXR) due to its epimerization to 3 alpha-epimer by hepatic metabolism. Journal of Steroid Biochemistry and Molecular Biology 2020, 202 (September), nestránkováno DOI: 10.1016/j.jsbmb.2020.105702.
Brynda, J.; Fanfrlík, J.; Hadzima, M.; Hánová, I.; Horn, M.; Houštecká, R.; Lepšík, M.; Majer, P.; Mareš, M.; Mertlíková-Kaiserová, H.; et al. Biomimetic Macrocyclic Inhibitors of Human Cathepsin D: Structure-Activity Relationship and Binding Mode Analysis. Journal of Medicinal Chemistry 2020, 63 (4), 1576-1596 DOI: 10.1021/acs.jmedchem.9b01351.
Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.
Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.
Báječný, M.; Beneš, J.; Czernek, J.; Dunlop, D.; Francová, P.; Groborz, O.; Heizer, T.; Hobza, P.; Hrubý, M.; Kolouchová, K.; et al. Chelating Polymers for Hereditary Hemochromatosis Treatment. Macromolecular Bioscience 2020, 20 (12), nestránkováno DOI: 10.1002/mabi.202000254.
Gálisová, A.; Groborz, O.; Hájek, M.; Hrubý, M.; Jirák, D.; Kolouchová, K.; Sedláček, O.; Sticová, E.; Švec, P.; Trousil, J.; et al. Implant-forming polymeric 19F MRI-tracer with tunable dissolution. Journal of Controlled Release 2020, 327 (November), 50-60 DOI: 10.1016/j.jconrel.2020.07.026.
Gálisová, A.; Groborz, O.; Hájek, M.; Hrubý, M.; Jirák, D.; Kolouchová, K.; Sedláček, O.; Sticová, E.; Švec, P.; Trousil, J.; et al. Implant-forming polymeric 19F MRI-tracer with tunable dissolution. Journal of Controlled Release 2020, 327 (November), 50-60 DOI: 10.1016/j.jconrel.2020.07.026.
Gálisová, A.; Groborz, O.; Hájek, M.; Hrubý, M.; Jirák, D.; Kolouchová, K.; Sedláček, O.; Sticová, E.; Švec, P.; Trousil, J.; et al. Implant-forming polymeric 19F MRI-tracer with tunable dissolution. Journal of Controlled Release 2020, 327 (November), 50-60 DOI: 10.1016/j.jconrel.2020.07.026.
Bušek, P.; Konvalinka, J.; Šedo, A.; Šimková, A. Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications. Biochimica et Biophysica Acta - Proteins and Proteomics 2020, 1868 (7), nestránkováno DOI: 10.1016/j.bbapap.2020.140409.
Bušek, P.; Konvalinka, J.; Šedo, A.; Šimková, A. Molecular recognition of fibroblast activation protein for diagnostic and therapeutic applications. Biochimica et Biophysica Acta - Proteins and Proteomics 2020, 1868 (7), nestránkováno DOI: 10.1016/j.bbapap.2020.140409.
Anania, M.; Jašík, J.; Jašíková, L.; Roithová, J.; Shcherbachenko, E.; Zelenka, J. Monoaurated vs. diaurated intermediates: causality or independence?. Chemical Science 2020, 11 (4), 980-988 DOI: 10.1039/c9sc05662a.
Barek, J.; Klouda, J.; Kočovský, P.; Nesměrák, K.; Schwarzova-Peckova, K. A novel voltammetric approach to the detection of primary bile acids in serum samples. Bioelectrochemistry 2020, 134 (August), nestránkováno DOI: 10.1016/j.bioelechem.2020.107539.
Bastien, G.; Císařová, I.; Dračínský, M.; Hurtado, C. Santos; Kaleta, J.; Mašát, M.; Rogers, C. T.; Rončević, I.; Štoček, J. Radek. Regular Two-Dimensional Arrays of Surface-Mounted Molecular Switches: Switching Monitored by UV-vis and NMR Spectroscopy. Journal of the American Chemical Society 2020, 142 (20), 9337-9351 DOI: 10.1021/jacs.0c01753.
Bursová, M.; Čabala, R.; Hložek, T.; Jelinek, I.; Štícha, M.; Tůma, P. Sensitive CE-MS method for monitoring of riociguat and desmethylriociguat levels in human serum. Electrophoresis 2020, 41 (18-19), 1564-1567 DOI: 10.1002/elps.202000135.
Brynda, J.; Das, V.; Dvořanová, J.; Džubák, P.; Anwar, S. El; Fábry, M.; Grüner, B.; Gurska, S.; Hajdúch, M.; Havránek, M.; et al. Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX. European Journal of Medicinal Chemistry 2020, 200 (August), nestránkováno DOI: 10.1016/j.ejmech.2020.112460.
Bartova, K.; Džubák, P.; Fleuti, M. Heidi; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Slavětínská, L. Poštová; Tichý, M.; Tloušťová, E. Synthesis and Biological Profiling of Pyrazolo-Fused 7-Deazapurine Nucleosides. Journal of Organic Chemistry 2020, 85 (16), 10539-10551 DOI: 10.1021/acs.joc.0c00928.
Fojta, M.; Havran, L.; Havranova-Vidlakova, P.; Hocek, M.; Krömer, M.; Sykorova, V.; Trefulka, M. Vicinal Diol-Tethered Nucleobases as Targets for DNA Redox Labeling with Osmate Complexes. Chembiochem : a European journal of chemical biology 2020, 21 (1-2), 171-180 DOI: 10.1002/cbic.201900388.
2018
Sabat, N.; Slavětínská, L. Poštová; Klepetářová, B.; Hocek, M. C-H Imidation of 7-Deazapurines. Acs Omega 2018, 3 (4), 4674-4678 DOI: 10.1021/acsomega.8b00520.
Sabat, N.; Slavětínská, L. Poštová; Klepetářová, B.; Hocek, M. C-H Imidation of 7-Deazapurines. Acs Omega 2018, 3 (4), 4674-4678 DOI: 10.1021/acsomega.8b00520.
Docekal, V.; Šimek, M.; Dračínský, M.; Vesely, J. Decarboxylative Organocatalytic Allylic Amination of Morita-Baylis-Hillman Carbamates. Chemistry-a European Journal 2018, 24 (51), 13441-13445 DOI: 10.1002/chem.201803677.
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