Publications

Bursová, M.; Čabala, R.; Hložek, T.; Jelinek, I.; Štícha, M.; Tůma, P. Sensitive CE-MS method for monitoring of riociguat and desmethylriociguat levels in human serum. Electrophoresis 2020, 41 (18-19), 1564-1567 DOI: 10.1002/elps.202000135.

Císařová, I.; Hara, S.; Kotora, M.; Topolovčan, N.; Tošner, Z. A Study of Polarization and Directing Effects of Unsymmetrical Alkynes Using Regioselective Pd-Catalyzed Bromoallylation. European Journal of Organic Chemistry 2020, 2020 (2), 234-240 DOI: 10.1002/ejoc.201901476.

Císařová, I.; Hara, S.; Kotora, M.; Topolovčan, N.; Tošner, Z. A Study of Polarization and Directing Effects of Unsymmetrical Alkynes Using Regioselective Pd-Catalyzed Bromoallylation. European Journal of Organic Chemistry 2020, 2020 (2), 234-240 DOI: 10.1002/ejoc.201901476.

Bartova, K.; Džubák, P.; Fleuti, M. Heidi; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Slavětínská, L. Poštová; Tichý, M.; Tloušťová, E. Synthesis and Biological Profiling of Pyrazolo-Fused 7-Deazapurine Nucleosides. Journal of Organic Chemistry 2020, 85 (16), 10539-10551 DOI: 10.1021/acs.joc.0c00928.

Bartova, K.; Džubák, P.; Fleuti, M. Heidi; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Slavětínská, L. Poštová; Tichý, M.; Tloušťová, E. Synthesis and Biological Profiling of Pyrazolo-Fused 7-Deazapurine Nucleosides. Journal of Organic Chemistry 2020, 85 (16), 10539-10551 DOI: 10.1021/acs.joc.0c00928.

Džubák, P.; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Pohl, R.; Tichý, M.; Yang, C. Synthesis, Photophysical Properties, and Biological Profiling of Benzothieno-Fused 7-Deazapurine Ribonucleosides. Journal of Organic Chemistry 2020, 85 (12), 8085-8101 DOI: 10.1021/acs.joc.0c00927.

Fojta, M.; Havran, L.; Havranova-Vidlakova, P.; Hocek, M.; Krömer, M.; Sykorova, V.; Trefulka, M. Vicinal Diol-Tethered Nucleobases as Targets for DNA Redox Labeling with Osmate Complexes. Chembiochem : a European journal of chemical biology 2020, 21 (1-2), 171-180 DOI: 10.1002/cbic.201900388.

Břehová, P.; Česnek, M.; Dračínský, M.; Chaloupecká, E.; Janeba, Z.; Mertlíková-Kaiserová, H.; Skácel, J.; Soto-Velasquez, M. P.; Tloušťová, E.; Watts, V. J. Acyclic nucleoside phosphonates with 2-aminothiazole base as inhibitors of bacterial and mammalian adenylate cyclases. European Journal of Medicinal Chemistry 2021, 222 (October 15 2021), nestránkováno.

Bricout, H.; Caronia, E.; Galia, A.; Tichá, I. Chena; Jindřich, J.; Léger, B.; Menuel, S.; Monflier, É.; Noël, S.; Ponchel, A.; et al. Asymmetric hydrogenation of ethyl pyruvate over aqueous dispersed Pt nanoparticles stabilized by a cinchonidine-functionalized β-cyclodextrin. Catalysis Communications 2021, 150 (February), nestránkováno.

Bricout, H.; Caronia, E.; Galia, A.; Tichá, I. Chena; Jindřich, J.; Léger, B.; Menuel, S.; Monflier, É.; Noël, S.; Ponchel, A.; et al. Asymmetric hydrogenation of ethyl pyruvate over aqueous dispersed Pt nanoparticles stabilized by a cinchonidine-functionalized β-cyclodextrin. Catalysis Communications 2021, 150 (February), nestránkováno.

Groborz, O.; Holubová, M.; Hromádková, J.; Hrubý, M.; Lobaz, V.; Loukotová, L.; Pechrová, Z.; Rabyk, M.; Štěpánek, P.; Trhlíková, O. Chemically modified glycogens: How they influence formation of amyloid fibrils?. Soft Matter 2021, 17 (6), 1614-1627.

Čihák, M.; Hurný, D.; Malečková, A.; Štuka, Č.; Tonar, Z.; Vejražka, M. "Desatero" akademického pedagoga. https://karlovkaonline.cz/wp-content/uploads/2021/04/UK_fond-desatero_www.pdf, 2021.

Bednářová, E.; Kotora, M.; Malatinec, Š.; Tanaka, H. Highly Enantioselective Ring-Opening of meso-Epoxides with O- and N-Nucleophiles Catalyzed by a Chiral Sc(III)/bipyridine Complex. European Journal of Organic Chemistry 2021, 2021 (8), 1249-1257.

Baszczyňski, O.; Císařová, I.; Flieger, M.; Kolařík, M.; Kucherak, O.; Procházková, E.; Stodůlková, E.; Tošner, Z. NMR Structure Elucidation of Naphthoquinones from Quambalaria cyanescens. Journal of Natural Products 2021, 84 (1), 46-55.

Gallardo, P. Güixens; Hocek, M.; Kraus, T.; Kuba, M.; Matyašovský, J.; Palágyi, A.; Pohl, R.; Tack, L. Nucleotides bearing aminophenyl- or aminonaphthyl-3-methoxychromone solvatochromic fluorophores for the enzymatic construction of DNA probes for the detection of protein-DNA binding. Organic and Biomolecular Chemistry 2021, 19 (45), 9966-9974.

Baszczyňski, O.; Gallardo, M. García; Procházková, E.; Šimon, P.; Tichotová, M. Phosphate-Based Self-Immolative Linkers for Tuneable Double Cargo Release. Chemistry - A European Journal 2021, 27 (50), 12763-12775.

Doleželová, E.; Downey, A. Michael; Hocek, M.; Nguyen, V. Hai; Pohl, R.; Rožánková, S.; Slapničková, M.; Tichý, M.; Tloušťová, E.; Zíková, A. Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides. Bioorganic and Medicinal Chemistry Letters 2021, 40 (May 15 2021), nestránkováno.

Doleželová, E.; Downey, A. Michael; Hocek, M.; Nguyen, V. Hai; Pohl, R.; Rožánková, S.; Slapničková, M.; Tichý, M.; Tloušťová, E.; Zíková, A. Synthesis and anti-trypanosomal activity of 3'-fluororibonucleosides derived from 7-deazapurine nucleosides. Bioorganic and Medicinal Chemistry Letters 2021, 40 (May 15 2021), nestránkováno.

Doleželová, E.; Džubák, P.; Gurská, S.; Hajdúch, M.; Hocek, M.; Krajczyk, A.; Milisavljević, N.; Perlíková, P.; Slavětínská, L. Poštová; Slapničková, M.; et al. Synthesis and Antitrypanosomal Activity of 6-Substituted 7-Methyl-7-deazapurine Nucleosides. ACS Infectious Diseases 2021, 7 (4), 917-926.

Hurný, D.; Malečková, A.; Štuka, Č.; Tonar, Z.; Vejražka, M. Ten evidence-based recommendations for higher education. Mefanet+ 2021: Cooperation on the effective use of technology in medical and healthcare education reflecting on the challenges of today, 2021, 13-13.

Čikoš, A.; Degač, M.; Gredičak, M.; Topolovčan, N. Chemoselective and Regioselective Synthesis of Spiroisoindolinone Indenes via an Intercepted Meyer–Schuster Rearrangement/Intramolecular Friedel–Crafts Alkylation Relay. Journal of Organic Chemistry 2022, 87 (5), 3712-3717.

Ausserlechner, M. J.; Dočekal, V.; Hagenbuchner, J.; Horváth, M.; Kaiser, N.; Kohoutová, K.; Mandal, R.; Obšil, T.; Obšilová, V.; Tekel, A.; et al. Lengthening the Guanidine–Aryl Linker of Phenylpyrimidinylguanidines Increases Their Potency as Inhibitors of FOXO3-Induced Gene Transcription. ACS Omega [online] 2022, 7 (38), 34632-34646.

Ausserlechner, M.; Dočekal, V.; Kohoutová, K.; Obšil, T.; Obšilová, V.; Tekel, A.; Veselý, J. Modulating FOXO3 transcriptional activity by low-molecular compounds. FEBS Open Bio [online], 2022, 12, 233-233.

Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.

Novotná, K.; Tenora, L.; Prchalová, E.; Paule, J.; Alt, J.; Veeravalli, V.; Lam, J.; Wu, Y.; Šnajdr, I.; Gori, S.; et al. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry 2023, 66 (22), 15493-15510.