Publications

Doleželová, E.; Džubák, P.; Gurská, S.; Hajdúch, M.; Hocek, M.; Krajczyk, A.; Milisavljević, N.; Perlíková, P.; Slavětínská, L. Poštová; Slapničková, M.; et al. Synthesis and Antitrypanosomal Activity of 6-Substituted 7-Methyl-7-deazapurine Nucleosides. ACS Infectious Diseases 2021, 7 (4), 917-926.

Konvalinka, J.; Kožíšek, M.; Kráľ, M.; Machara, A.; Majer, P.; Radilová, K.; Reiberger, R. Synthesis and In Vitro Evaluation of C-7 and C-8 Luteolin Derivatives as Influenza Endonuclease Inhibitors, 2021.

Císařová, I.; Henriksson, E.; Kamlar, M.; Malo, M.; Sunden, H. Synthesis of cis-Oriented Vicinal Diphenylethylenes through a Lewis Acid-Promoted Annulation of Oxotriphenylhexanoates. Journal of Organic Chemistry 2021, 86 (13), 8660-8671.

Bažíková, E.; Císařová, I.; Jagtap, P. Ramling; Matoušová, E.; Nechaev, A.; Neumannová, J. Synthesis of fused 1,2-naphthoquinones with cytotoxic activity using a one-pot three-step reaction. Organic and Biomolecular Chemistry 2021, 19 (15), 3434-3440.

Bakhanovich, O.; Beier, P.; Khutorianskyi, V.; Motornov, V. Synthesis of N-perfluoroalkyl-3,4-disubstituted pyrroles by rhodium-catalyzed transannulation of N-fluoroalkyl-1,2,3-triazoles with terminal alkynes. Beilstein Journal of Organic Chemistry 2021, 17 (February 18 2021), 504-510.

Bursová, M.; Čabala, R.; Hložek, T.; Jelinek, I.; Štícha, M.; Tůma, P. Sensitive CE-MS method for monitoring of riociguat and desmethylriociguat levels in human serum. Electrophoresis 2020, 41 (18-19), 1564-1567 DOI: 10.1002/elps.202000135.

Baszczynski, O.; Cigáň, M.; Filo, J.; Prochazkova, E. Sterically-Controlled Self-Immolation in Phosphoramidate Linkers Triggered by Light. European Journal of Organic Chemistry 2020, 2020 (7), 897-906 DOI: 10.1002/ejoc.201901882.

Císařová, I.; Hara, S.; Kotora, M.; Topolovčan, N.; Tošner, Z. A Study of Polarization and Directing Effects of Unsymmetrical Alkynes Using Regioselective Pd-Catalyzed Bromoallylation. European Journal of Organic Chemistry 2020, 2020 (2), 234-240 DOI: 10.1002/ejoc.201901476.

Brynda, J.; Das, V.; Dvořanová, J.; Džubák, P.; Anwar, S. El; Fábry, M.; Grüner, B.; Gurska, S.; Hajdúch, M.; Havránek, M.; et al. Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX. European Journal of Medicinal Chemistry 2020, 200 (August), nestránkováno DOI: 10.1016/j.ejmech.2020.112460.

Bartova, K.; Džubák, P.; Fleuti, M. Heidi; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Slavětínská, L. Poštová; Tichý, M.; Tloušťová, E. Synthesis and Biological Profiling of Pyrazolo-Fused 7-Deazapurine Nucleosides. Journal of Organic Chemistry 2020, 85 (16), 10539-10551 DOI: 10.1021/acs.joc.0c00928.

Džubák, P.; Gurska, S.; Hajdúch, M.; Hocek, M.; Pavliš, P.; Pohl, R.; Tichý, M.; Yang, C. Synthesis, Photophysical Properties, and Biological Profiling of Benzothieno-Fused 7-Deazapurine Ribonucleosides. Journal of Organic Chemistry 2020, 85 (12), 8085-8101 DOI: 10.1021/acs.joc.0c00927.

Bakhanovich, O.; Beier, P. Synthesis, Stability and Reactivity of alpha-Fluorinated Azidoalkanes. Chemistry - A European Journal 2020, 26 (4), 773-782 DOI: 10.1002/chem.201903627.

Ivancova, I.; Pohl, R.; Hubalek, M.; Hocek, M. Squaramate-Modified Nucleotides and DNA for Specific Cross-Linking with Lysine-Containing Peptides and Proteins. Angewandte Chemie-International Edition 2019, 58 (38), 13345-13348 DOI: 10.1002/anie.201906737.

Markos, A.; Voltrova, S.; Motornov, V.; Tichy, D.; Klepetářová, B.; Beier, P. Stereoselective Synthesis of (Z)-beta-Enamido Triflates and Fluorosulfonates from N-Fluoroalkylated Triazoles. Chemistry-a European Journal 2019, 25 (32), 7640-7644 DOI: 10.1002/chem.201901632.

Malnuit, V.; Smolen, S.; Tichý, M.; Slavětínská, L. Poštová; Hocek, M. Synthesis of Cyclic and Acyclic Nucleoside Phosphonates and Sulfonamides Derived from 6-(Thiophen-2-yl)-7-fluoro-7-deazapurine. European Journal of Organic Chemistry 2019, 2019 (31-32), 5409-5423 DOI: 10.1002/ejoc.201900509.

Krömer, M.; Bartova, K.; Raindlová, V.; Hocek, M. Synthesis of Dihydroxyalkynyl and Dihydroxyalkyl Nucleotides as Building Blocks or Precursors for Introduction of Diol or Aldehyde Groups to DNA for Bioconjugations. Chemistry-a European Journal 2018, 24 (46), 11890-11894 DOI: 10.1002/chem.201802282.

Andris, E.; Navrátil, R.; Jašík, J.; Sabenya, G.; Costas, M.; Srnec, M.; Roithová, J. Spin-State-Controlled Photodissociation of Iron(III) Azide to an Iron(V) Nitride Complex. Angewandte Chemie-International Edition 2017, 56 (45), 14057-14060 DOI: 10.1002/anie.201707420.

A. Downey, M.; Pohl, R.; Roithová, J.; Hocek, M. Synthesis of Nucleosides through Direct Glycosylation of Nucleobases with 5-O-Monoprotected or 5-Modified Ribose: Improved Protocol, Scope, and Mechanism. Chemistry-a European Journal 2017, 23 (16), 3910-3917 DOI: 10.1002/chem.201604955.

Kaiser, R. P.; Mosinger, J.; Císařová, I.; Kotora, M. Synthesis of selectively 4-substituted 9,9 '-spirobifluorenes and modulation of their photophysical properties. Organic & Biomolecular Chemistry 2017, 15 (33), 6913-6920 DOI: 10.1039/c7ob01319a.

Dziuba, D.; Pospíšil, P.; Matyašovský, J.; Brynda, J.; Nachtigallová, D.; Rulíšek, L.; Pohl, R.; Hof, M.; Hocek, M. Solvatochromic fluorene-linked nucleoside and DNA as color-changing fluorescent probes for sensing interactions. Chem. Sci. 2016, 7 (9), 5775-5785 DOI: 10.1039/C6SC02548J.

Machara, A.; Lux, V.; Kožíšek, M.; Šašková, K. Grantz; Štěpánek, O.; Kotora, M.; Parkan, K.; Pávová, M.; Glass, B.; Sehr, P.; et al. Specific Inhibitors of HIV Capsid Assembly Binding to the C-Terminal Domain of the Capsid Protein: Evaluation of 2-Arylquinazolines as Potential Antiviral Compounds. Journal of Medicinal Chemistry 2016, 59 (2), 545-558 DOI: 10.1021/acs.jmedchem.5b01089.

Andris, E.; Jašík, J.; Gómez, L.; Costas, M.; Roithová, J. Spectroscopic Characterization and Reactivity of Triplet and Quintet Iron(IV) Oxo Complexes in the Gas Phase. Angewandte Chemie International Edition 2016, 55 (11), 3637-3641 DOI: 10.1002/anie.201511374.

Humpl, M.; Tauchman, J.; Topolovčan, N.; Kretschmer, J.; Hessler, F.; Císařová, I.; Kotora, M.; Vesely, J. Stereoselective Synthesis of Ezetimibe via Cross-Metathesis of Homoallylalcohols and α-Methylidene-β-Lactams. The Journal of Organic Chemistry 2016, 81 (17), 7692-7699 DOI: 10.1021/acs.joc.6b01406.

Mikušek, J.; Matouš, P.; Matoušová, E.; Janoušek, M.; Kuneš, J.; Pour, M. Substrate Control in the Gold(I)-Catalyzed Cyclization of β - Propargylamino Acrylic Esters and Further Transformations of the Resultant Dihydropyridines. Advanced Synthesis & Catalysis 2016, 358 (18), 2912-2922 DOI: 10.1002/adsc.201600412.

Benkovics, G.; Hodek, O.; Havlikova, M.; Bosakova, Z.; Coufal, P.; Malanga, M.; Fenyvesi, E.; Darcsi, A.; Beni, S.; Jindřich, J. Supramolecular structures based on regioisomers of cinnamyl-α-cyclodextrins – new media for capillary separation techniques. Beilstein Journal of Organic Chemistry 2016, 12, 97-109 DOI: 10.3762/bjoc.12.11.