Publications

Jansa, P.; Císařová, I.; Matoušová, E. Oxidative Cleavage and Ring Reconstruction for the Synthesis of Amaryllidaceae Alkaloid Analogues. European Journal of Organic Chemistry 2024, 27 (3).

Baris, N.; Dračínský, M.; Tarábek, J.; Filgas, J.; Slavíček, P.; Ludvíková, L.; Boháčová, S.; Slanina, T.; Klepetářová, B.; Beier, P. Photocatalytic Generation of Trifluoromethyl Nitrene for Alkene Aziridination. Angewandte Chemie - International Edition 2024, 63 (2).

Hadzima, M.; Faucher, F. F.; Blažková, K.; Yim, J. J.; Guerra, M.; Chen, S.; Woods, E. C.; Park, K. Wan; Šácha, P.; Šubr, V.; et al. Polymer-Tethered Quenched Fluorescent Probes for Enhanced Imaging of Tumor-Associated Proteases. ACS Sensors 2024, 9 (7), 3720-3729.

Lebedinskiy, K.; Barvík, I.; Tošner, Z.; Císařová, I.; Jindřich, J.; Hrdina, R. Spatial arrangements of cyclodextrin host–guest complexes in solution studied by ¹³C NMR and molecular modelling. Beilstein Journal of Organic Chemistry 2024, 20 (February), 331-335.

Nosek, V.; Míšek, J. Sulfinamide Crossover Reaction. Journal of Organic Chemistry 2024, 89 (11), 7927-7932.

Fleuti, M. Heidi; Quirante, T. Sanchez; Slavětínská, L. Poštová; Tloušťová, E.; Tichý, M.; Gurská, S.; Džubák, P.; Hajdúch, M.; Hocek, M. Synthesis and Biological Profiling of Quinolino-Fused 7-Deazapurine Nucleosides. ACS Omega 2024, 9 (18), 20557-20570.

Topolovčan, N.; Kotora, M. Synthesis of 1,2-Disubstituted Cyclopentadienes and Their Application. In Metallocenes in Regio- and Stereoselective Synthesis; Metallocenes in Regio- and Stereoselective Synthesis; Springer, 2024; pp 19-46.

Dočekal, V.; Melaimi, M.; Petrželová, S.; Veselý, J.; Yan, X.; Bertrand, G. Synthesis of enantiopure 1,2,3-triazolylidene-type mesoionic carbene (MIC) conjugate acids featuring a rigid bicyclic scaffold. Organic Chemistry Frontiers 2024, 11 (8), 2178-2181.

Janecký, L.; Klepetářová, B.; Beier, P. Transformation of 5-acylated N-fluoroalkyl-1,2,3-triazoles to trifluoromethylated ring-fused isoquinolines, 1,3-oxazines, and 1,3-oxazin-6-ones via ketenimines. RSC Advances 2024, 14 (37), 26938-26942.

Osifová, Z.; Kalvoda, T.; Galgonek, J.; Culka, M.; Vondrášek, J.; Bouř, P.; Bednárová, L.; Andrushchenko, V.; Dračínský, M.; Rulíšek, L. What are the minimal folding seeds in proteins? Experimental and theoretical assessment of secondary structure propensities of small peptide fragments. Chemical Science 2024, 15 (2), 594-608.

Vopálenská, A.; Dočekal, V.; Petrželová, S.; Císařová, I.; Veselý, J. Access to Spirooxindole-Fused Cyclopentanes via a Stereoselective Organocascade Reaction Using Bifunctional Catalysis. Journal of Organic Chemistry 2023, 88 (12), 7724-7735.

Jestřábová, I.; Slavětínská, L. Poštová; Hocek, M. Arylethynyl- or Alkynyl-Linked Pyrimidine and 7-Deazapurine 2′-Deoxyribonucleoside 3′-Phosphoramidites for Chemical Synthesis of Hypermodified Hydrophobic Oligonucleotides. ACS Omega 2023, 8 (42), 39447-39453.

Ulč, J.; Jacko, J.; Císařová, I.; Pospíšil, L.; Nečas, D.; Kotora, M. Catalytic C−C/C−H Bond Activation Relay for Synthesis of Fluorescent Naphthoquinolizinium Salts. European Journal of Organic Chemistry 2023, 26 (18).

Fadeev, A.; Kotora, M. Catalytic vs. uncatalyzed [2+2] photocycloadditions of quinones with alkynes. Organic and Biomolecular Chemistry 2023, 21 (30), 6174-6179.

Brunderová, M.; Krömer, M.; Vlková, M.; Hocek, M. Chloroacetamide-Modified Nucleotide and RNA for Bioconjugations and Cross-Linking with RNA-Binding Proteins. Angewandte Chemie - International Edition 2023, 62 (7).

Martínek, M.; Ludvíková, L.; Šranková, M.; Navrátil, R.; Muchová, L.; Huzlík, J.; Vítek, L.; Klán, P.; Šebej, P. Common xanthene fluorescent dyes are visible-light activatable CO-releasing molecules. Organic and Biomolecular Chemistry 2023, 21 (1), 93-97.

Jabczun, M.; Nosek, V.; Míšek, J. Complementary strategies for synthesis of sulfinamides from sulfur-based feedstock. Organic and Biomolecular Chemistry 2023, 21 (14), 2950-2954.

Orosz, J. Máté; Ujj, D.; Kasal, P.; Benkovics, G.; Bálint, E. Continuous flow synthesis of 6-monoamino-6-monodeoxy-β-cyclodextrin. Beilstein Journal of Organic Chemistry 2023, 19 (Mar 9 2023), 294-302.

Cadart, T. Christophe; Gläsel, T.; Císařová, I.; Gyepes, R.; Nečas, D.; Hapke, M.; Kotora, M. Cyclotrimerization Approach to Symmetric [9]Helical Indenofluorenes: Diverting Cyclization Pathways. Chemistry - A European Journal 2023, 29 (58).

Prener, L.; Baszczyňski, O.; Kaiser, M. Maxmilian; Dračínský, M.; Stepan, G.; Lee, Y. - J.; Brumshtein, B.; Yu, H.; Jansa, P.; Lansdon, E. B.; et al. Design and Synthesis of Novel HIV-1 NNRTIs with Bicyclic Cores and with Improved Physicochemical Properties. Journal of Medicinal Chemistry 2023, 66 (3), 1761-1777.

Skácel, J.; Djukic, S.; Baszczyňski, O.; Kalčic, F.; Bílek, T.; Chalupský, K.; Kozák, J.; Dvořáková, A.; Tloušťová, E.; Kráľová, Z.; et al. Design, Synthesis, Biological Evaluation, and Crystallographic Study of Novel Purine Nucleoside Phosphorylase Inhibitors. Journal of Medicinal Chemistry 2023, 66 (10), 6652-6681.

Novotná, K.; Tenora, L.; Prchalová, E.; Paule, J.; Alt, J.; Veeravalli, V.; Lam, J.; Wu, Y.; Šnajdr, I.; Gori, S.; et al. Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery. Journal of Medicinal Chemistry 2023, 66 (22), 15493-15510.

Holovko-Kamoshenkova, O. M.; Slivka, M. V.; Hrdina, R.; Baumer, V. N.; Korol, N. I.; Sokolenko, L. V.; Lendel, V. G. An Efficient Catalyst-Free Direct Approach to 5-Polyfluoroalkyl-1,2,4-triazole-3-thiones. Synthesis 2023, 55 (08), 1221-1226.

Spampinato, A.; Kužmová, E.; Pohl, R.; Sýkorová, V.; Vrábel, M.; Kraus, T.; Hocek, M. trans-Cyclooctene- and Bicyclononyne-Linked Nucleotides for Click Modification of DNA with Fluorogenic Tetrazines and Live Cell Metabolic Labeling and Imaging. Bioconjugate Chemistry 2023, 34 (4), 772-780.

Belhajová, M.; Vícha, A.; Burgert, L.; Brožková, I.; Michaličková, L.; Hrdina, R.; Moravec, T.; Netuka, D.; Musil, Z.; Hrdina, R. En route to local glioblastoma treatment with temozolomide doped hyaluronan fibres: formulation and in vitro cell studies. RSC Medicinal Chemistry 2023, 14 (9), 1662-1666.